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Catalog No. Product Name Information Product Use Citations Product Validations
S8141 Cl-amidine Cl-amidine is an irreversible pan-peptidylarginine deiminase (PAD) inhibitor with IC50 values of 5.9 ± 0.3 μM, 0.8 ± 0.3 μM, 6.2 ± 1.0 μM for PAD4, PAD1 and PAD3, respectively. Cl-amidine induces apoptosis.
Immunity, 2025, S1074-7613(25)00069-X
Cell Rep, 2025, 44(2):115226
Nat Commun, 2024, 15(1):8663
S7803 GSK484 HCl GSK484 HCl, a benzoimidazole derivative, is a selective and reversible inhibitor of peptidylarginine deiminase 4 (PAD4) with IC50 of 50 nM in the absence of Calcium.
Cancer Cell, 2025, 43(1):69-85.e11
J Exp Clin Cancer Res, 2024, 43(1):319
Eur J Pharmacol, 2024, S0014-2999(24)00322-4
S9644 BMS-P5 BMS-P5, a potent selective pharmacological inhibitor of PAD4, is used to evaluate the effect of PAD4 inhibition on multiple myeloma (MM)-induced neutrophil extracellular trap (NET) formation.
S7802 GSK199 GSK199 is a selective inhibitor of PAD4 with IC50 of 200 nM in the absence of calcium.
S8141 Cl-amidine Cl-amidine is an irreversible pan-peptidylarginine deiminase (PAD) inhibitor with IC50 values of 5.9 ± 0.3 μM, 0.8 ± 0.3 μM, 6.2 ± 1.0 μM for PAD4, PAD1 and PAD3, respectively. Cl-amidine induces apoptosis.
Immunity, 2025, S1074-7613(25)00069-X
Cell Rep, 2025, 44(2):115226
Nat Commun, 2024, 15(1):8663
S7803 GSK484 HCl GSK484 HCl, a benzoimidazole derivative, is a selective and reversible inhibitor of peptidylarginine deiminase 4 (PAD4) with IC50 of 50 nM in the absence of Calcium.
Cancer Cell, 2025, 43(1):69-85.e11
J Exp Clin Cancer Res, 2024, 43(1):319
Eur J Pharmacol, 2024, S0014-2999(24)00322-4
S9644 BMS-P5 BMS-P5, a potent selective pharmacological inhibitor of PAD4, is used to evaluate the effect of PAD4 inhibition on multiple myeloma (MM)-induced neutrophil extracellular trap (NET) formation.
S7802 GSK199 GSK199 is a selective inhibitor of PAD4 with IC50 of 200 nM in the absence of calcium.

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Tags: PAD inhibitor|PAD agonist|PAD activator|PAD inducer|PAD antagonist|PAD signaling pathway|PAD assay kit